SCHEMBL5526316

SCHEMBL5526316

Nc1nc(-c2ccccc2)ccc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.50
MAP2K3 P46734 1/20 0.49
MEN1 O00255 6/20 0.48
KMT2A Q03164 6/20 0.48
RAB9A P51151 1/20 0.48
MAPT P10636 3/20 0.47
LMNA P02545 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK10 P53779 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ADORA2A P29274 6/20 0.47
ADORA1 P30542 6/20 0.47
HSP90AA1 P07900 2/20 0.47
AURKA O14965 1/20 0.47
PRKACA P17612 1/20 0.47
FTO Q9C0B1 1/20 0.45
EGLN1 Q9GZT9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053052 0.78 MAP2K3 (0.56) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL21857026 0.75 MAP2K3 (0.58) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL28247990 0.75 ASIC3 (0.50) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL1360818 0.75 ALDH1A1 (0.59) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL27807144 0.75 ALDH1A1 (0.64) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL14917463 0.73 MEN1 (0.62) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL20472126 0.72 ADORA2A (0.48) RAB9AMAPTCYP1A2SMN1; SMN2ADORA2A
SCHEMBL8077324 0.72 ASIC3 (0.47) ASIC3MAP2K3MEN1KMT2ARAB9A
SCHEMBL19009938 0.72 TDO2 (0.45) MEN1KMT2ARAB9ACYP1A2FTO
SCHEMBL29106081 0.72 FTO (0.62) MAP2K3MEN1KMT2ARAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814888-A1 AZABENZOXAZOLES FOR THE TREATMENT OF CNS DISORDERS Pfizer Products Incorporated (US) 2007-08-08 EP disclosed
US-20060173179-A1 Azabenzoxazoles for the treatment of CNS disorders PFIZER INC 2006-08-03 US disclosed
WO-2006051394-A1 AZABENZOXAZOLES FOR THE TREATMENT OF CNS DISORDERS PFIZER PRODUCTS INC. (US) 2006-05-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173179-A1 Azabenzoxazoles for the treatment of CNS disorders CHRNA7, CHRNA5, CHRNA10 ASIC3 2913/4885MAP2K3 2960/4885MEN1 3862/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.