SCHEMBL5527997

SCHEMBL5527997

CCCCOC(=O)C(C(=O)O)C1CNC(c2ccc(C#N)cc2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.37
ALOX5 P09917 1/20 0.37
PPARG P37231 1/20 0.37
KCNH2 Q12809 1/20 0.37
MGLL Q99685 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
DPP4 P27487 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
PGR P06401 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HIF1A Q16665 1/20 0.33
CTSG P08311 1/20 0.33
CMA1 P23946 1/20 0.33
NOD2 Q9HC29 1/20 0.33
NOD1 Q9Y239 1/20 0.33
HRH2 P25021 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5530482 0.82 GPR119 (0.34) KCNH2L3MBTL1
SCHEMBL5527993 0.75 NOD2 (0.36) KCNH2MGLLL3MBTL1DPP4ALDH1A1
SCHEMBL1076478 0.68 CPN1 (0.36) ALDH1A1ITGB3ITGA2B
SCHEMBL7401485 0.67 CPN1 (0.41) ALDH1A1ITGB3ITGA2B
SCHEMBL3495579 0.66 KDM1A (0.38) KCNH2L3MBTL1PGR
SCHEMBL3495575 0.66 KDM1A (0.38) KCNH2L3MBTL1PGR
SCHEMBL3495572 0.66 KDM1A (0.38) KCNH2L3MBTL1PGR
SCHEMBL3496533 0.66 KDM1A (0.38) KCNH2L3MBTL1PGR
SCHEMBL3496531 0.66 KDM1A (0.38) KCNH2L3MBTL1PGR
SCHEMBL7529709 0.66 ACACB (0.46) MGLLDPP4ALDH1A1CTSGCMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804793-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047195-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed