SCHEMBL5528030

SCHEMBL5528030

O=CC(Br)(c1ccccc1)c1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 2/20 0.43
MAPK1 P28482 1/20 0.42
KIF11 P52732 1/20 0.40
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP1B1 Q16678 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
G6PD P11413 1/20 0.34
AKR1C3 P42330 1/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1414647 0.91 ESR1 (0.41) ALDH1A1TDP1MAPK1CA1CA2
SCHEMBL10538145 0.82 ALDH1A1 (0.43) ALDH1A1TDP1MAPK1KIF11CA1
SCHEMBL21495110 0.80 KIF11 (0.43) ALDH1A1MAPK1KIF11CA1CA2
SCHEMBL4015306 0.80 KCNN4 (0.50) ALDH1A1KIF11MEN1KMT2AKCNN4
SCHEMBL8796837 0.80 KIF11 (0.43) MAPK1KIF11MEN1KMT2ASMN1; SMN2
SCHEMBL5255832 0.80 ESR1 (0.59) ALDH1A1TDP1KIF11CA1CA2
SCHEMBL6629671 0.78 KIF11 (0.41) ALDH1A1TDP1MAPK1KIF11MAOA
SCHEMBL17941356 0.75 ALDH1A1 (0.53) ALDH1A1TDP1MAPK1KIF11CA1
SCHEMBL3083376 0.75 ALDH1A1 (0.53) ALDH1A1TDP1MAPK1KIF11CA1
SCHEMBL3956177 0.75 ALDH1A1 (0.53) ALDH1A1TDP1MAPK1KIF11CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748993-A1 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2007-02-07 EP disclosed
WO-2005116000-A1 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2005-12-08 WO disclosed
EP-1581214-A1 4,5-DIARYLTHIAZOLE DERIVATIVES AS CB-1 LIGANDS Astrazeneca AB (SE) 2005-10-05 EP disclosed
WO-2004058255-A1 4, 5-DIARYLTHIAZOLE DERIVATIVES AS CB-1 LIGANDS ASTRAZENECA AB (SE) 2004-07-15 WO disclosed