SCHEMBL5533438

SCHEMBL5533438

CS(=O)(=O)N(CCCc1ccc(C#N)cc1)CCN1CC2CN(CCOC(N)=O)CC(C1)O2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.38
DRD4 P21917 3/20 0.38
HTR2A P28223 3/20 0.38
HRH1 P35367 3/20 0.38
OPRM1 P35372 3/20 0.38
KCNH2 Q12809 3/20 0.38
CYP19A1 P11511 3/20 0.35
DRD2 P14416 4/20 0.35
DRD3 P35462 4/20 0.35
CACNA1F O60840 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
DRD1 P21728 2/20 0.35
DRD5 P21918 2/20 0.35
HRH2 P25021 2/20 0.35
ADRA1D P25100 2/20 0.35
HTR7 P34969 2/20 0.35
ADRA1A P35348 2/20 0.35
ADRA1B P35368 2/20 0.35
HTR6 P50406 2/20 0.35
CACNA1D Q01668 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5534239 0.88 KCNH2 (0.43) HRH1KCNH2HRH2HRH3MEN1
SCHEMBL4505273 0.83 HRH1 (0.37) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL5116804 0.83 KCNH2 (0.42) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4516179 0.83 KCNH2 (0.47) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4513667 0.83 OPRM1 (0.40) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4508018 0.82 GPR119 (0.40) HTR1ADRD4HTR2AHRH1OPRM1
Hydrochloric Acid SCHEMBL4521680 0.82 KCNH2 (0.36) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4512005 0.82 KCNH2 (0.36) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4669141 0.82 OPRM1 (0.44) HTR1ADRD4HTR2AHRH1OPRM1
SCHEMBL4523088 0.81 KCNH2 (0.37) HTR1ADRD4HTR2AHRH1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765831-A1 NOVEL OXABISPIDINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CARDIAC ARRHYTHMIAS AstraZeneca AB (SE) 2007-03-28 EP claimed
WO-2005123747-A1 NOVEL OXABISPIDINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2005-12-29 WO claimed