SCHEMBL5538112

SCHEMBL5538112

CCc1ccc(C(=O)NC2=NCC3=CN(S(=O)(=O)c4ccc5c(c4)CN(C(=O)C(F)(F)F)CC5)CCC3=N2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
MAPT P10636 2/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
OPRK1 P41145 3/20 0.36
MOGAT2 Q3SYC2 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
ADCY8 P40145 1/20 0.34
ADCY1 Q08828 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HTT P42858 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5538108 0.79 PKM (0.42) PKMMAPTESR1ESR2OPRK1
SCHEMBL5545059 0.79 ALDH1A1 (0.46) NPC1RAB9AHTT
SCHEMBL3530530 0.73 PKM (0.46) PKMMAPTESR1ESR2OPRK1
SCHEMBL5546201 0.72 ABL1 (0.40) HDAC6HTT
SCHEMBL5546901 0.72 ALDH1A1 (0.51) PKMMAPT
SCHEMBL5548489 0.71 TUBB4A (0.50) MAPTNPC1RAB9A
SCHEMBL5540390 0.68 RAB9A (0.35) PKMMAPTOPRK1NPC1RAB9A
SCHEMBL11477876 0.67 ESR1 (0.67) PKMESR1ESR2
Dimethylamine SCHEMBL6529354 0.67 ESR1 (0.62) PKMESR1ESR2HDAC6
SCHEMBL8277232 0.66 ESR1 (0.65) PKMESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed