SCHEMBL5540285

SCHEMBL5540285

O=C(NC1=NCC2=CN(S(=O)(=O)Cc3ccccc3)CCC2=N1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.39
NPC1 O15118 4/20 0.39
ALDH1A1 P00352 2/20 0.39
GPR183 P32249 1/20 0.39
CXCR2 P25025 1/20 0.38
MAPT P10636 1/20 0.38
SLC6A12 P48065 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
MCHR1 Q99705 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
TNF P01375 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
MAPK1 P28482 1/20 0.36
ABL1 P00519 1/20 0.35
SRC P12931 1/20 0.35
CHRM4 P08173 1/20 0.35
FKBP1A P62942 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540370 0.72 MAPT (0.41) RAB9ANPC1ALDH1A1MAPTKMT2A
SCHEMBL5543018 0.66 ALDH1A1 (0.43) RAB9ANPC1ALDH1A1MAPTKMT2A
SCHEMBL2919112 0.65 GPR183 (0.41) RAB9ANPC1ALDH1A1GPR183CXCR2
SCHEMBL3532982 0.64 CYP1A2 (0.52) RAB9ANPC1ALDH1A1GPR183MAPT
SCHEMBL2921797 0.64 NTRK1 (0.42) RAB9ANPC1ALDH1A1GPR183CXCR2
SCHEMBL2918827 0.63 CCNA2 (0.58)
SCHEMBL12310177 0.58 RAB9A (0.73) RAB9ANPC1ALDH1A1CXCR2MAPT
SCHEMBL4783063 0.57 MEN1 (0.86) RAB9ANPC1ALDH1A1MAPTKMT2A
SCHEMBL30616676 0.57 GPR183 (0.52) RAB9ANPC1GPR183KMT2AMAPK1
SCHEMBL5230740 0.57 HDAC6 (0.72) RAB9ANPC1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed