SCHEMBL5543566

SCHEMBL5543566

CC(C)c1nc(NCCCN2CCOCC2)c2n[nH]c(=O)n2c1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.52
TP53 P04637 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
ACP1 P24666 3/20 0.49
KDM4E B2RXH2 5/20 0.48
KMT2A Q03164 4/20 0.48
POLB P06746 3/20 0.48
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 3/20 0.48
MAPT P10636 2/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
TLR9 Q9NR96 4/20 0.46
GAA P10253 2/20 0.45
NPC1 O15118 2/20 0.45
LMNA P02545 2/20 0.45
RAB9A P51151 2/20 0.45
GLA P06280 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545608 0.85 MAPK1 (0.51) MAPK1TP53ALOX15TSHRACP1
SCHEMBL5548577 0.84 GAA (0.45) MAPK1TP53ALOX15TSHRACP1
SCHEMBL5549356 0.77 ALDH1A1 (0.55) MAPK1TP53ALOX15TSHRACP1
SCHEMBL5548536 0.76 GAA (0.47) MAPK1TP53ALOX15TSHRACP1
SCHEMBL5548924 0.75 ADORA1 (0.54) MAPK1TSHRPOLBALDH1A1MAPT
SCHEMBL5550115 0.73 GAA (0.45) MAPK1TP53ALOX15TSHRACP1
SCHEMBL3526664 0.69 GAA (0.45) MAPK1TP53ALOX15TSHRKDM4E
SCHEMBL7238360 0.66 KDM4E (0.62) MAPK1TP53ALOX15TSHRACP1
SCHEMBL6135962 0.66 ACP1 (0.43) MAPK1TP53ALOX15TSHRACP1
SCHEMBL10367734 0.65 KDM4E (0.57) MAPK1TP53ALOX15TSHRACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed