SCHEMBL5545154

SCHEMBL5545154

C[C@H](Nc1ccc(Br)cc1C(=O)c1ccccc1F)C(N)=O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
MAPT P10636 4/20 0.41
ALDH1A1 P00352 6/20 0.41
CTSL P07711 2/20 0.40
GSTA1 P08263 1/20 0.40
MAP2K2 P36507 1/20 0.39
MAP2K1 Q02750 1/20 0.39
MAPK1 P28482 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DGAT1 O75907 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1198598 0.81 TP53 (0.59) TP53MAPTALDH1A1MAPK1MEN1
SCHEMBL5583501 0.78 TP53 (0.56) TP53MAPTALDH1A1MAPK1MEN1
SCHEMBL1198846 0.78 TP53 (0.55) TP53MAPTALDH1A1CTSLGSTA1
SCHEMBL14998701 0.77 TP53 (0.57) TP53MAPTALDH1A1GSTA1MAPK1
SCHEMBL1198848 0.75 TP53 (0.61) TP53MAPTALDH1A1MAPK1L3MBTL1
SCHEMBL638047 0.74 MAPT (0.63) TP53MAPTALDH1A1CTSLGSTA1
SCHEMBL30375142 0.74 MAPT (0.63) TP53MAPTALDH1A1CTSLGSTA1
SCHEMBL30317493 0.74 MEN1 (0.53) MAPTALDH1A1MEN1KMT2ANPC1
SCHEMBL8586004 0.73 TP53 (0.62) TP53MAPTALDH1A1GSTA1MAPK1
SCHEMBL638831 0.73 TP53 (0.62) TP53MAPTALDH1A1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812112-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2007-08-01 EP disclosed
WO-2006044753-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-04-27 WO disclosed