SCHEMBL5545694

SCHEMBL5545694

Cc1cccc(C)c1N(c1c(C)cccc1C)P(N)(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.42
CD44 P16070 1/20 0.39
CYP3A4 P08684 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
ALDH1A1 P00352 4/20 0.33
TSHR P16473 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33
CA9 Q16790 2/20 0.33
PIK3CA P42336 1/20 0.33
HPGD P15428 1/20 0.33
ACHE P22303 1/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTR5A P47898 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8365536 0.77 ALDH1A1 (0.39) MAPTCD44CYP1A2CYP2A6ALDH1A1
O-Xylene SCHEMBL17338002 0.69 TSHR (0.62) MAPTCD44CYP3A4TDP1CYP1A2
Piperazine SCHEMBL329108 0.69 ADRB1 (0.39) CYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL12902950 0.66 CYP1A2 (0.47) MAPTCD44CYP3A4TDP1CYP1A2
SCHEMBL18509851 0.65 CD44 (0.52) CD44CYP3A4TDP1CYP1A2CYP2A6
SCHEMBL7029367 0.65 TSHR (0.44) MAPTCYP3A4TDP1ALDH1A1TSHR
SCHEMBL1726840 0.64 CYP2A6 (0.45) MAPTCD44TDP1CYP1A2CYP2A6
SCHEMBL1107763 0.64 CYP2A6 (0.45) MAPTCD44TDP1CYP1A2CYP2A6
SCHEMBL96680 0.64 HTT (0.48) MAPTCYP3A4TDP1CYP1A2ALDH1A1
SCHEMBL16776729 0.63 CD44 (0.72) CD44CYP3A4TDP1CYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112314-B1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GEN ELECTRIC (US) 2007-07-04 EP disclosed
EP-1131378-B1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GEN ELECTRIC (US) 2005-02-23 EP disclosed
US-6569929-B2 Containing thermoplastic resins GENERAL ELECTRIC COMPANY 2003-05-27 US disclosed
EP-1144498-B1 FLAME RETARDANT POLYMER BLENDS, AND METHOD FOR MAKING GEN ELECTRIC (US) 2002-10-09 EP disclosed
US-6433046-B1 MIXTURE WITH THERMOPLASTIC RESIN AND FLAME RETARDANT; COMPUTER HOUSINGS, PANELS, APPLIANCES, AUTOMOBILES, SPORTS EQUIPMENT; MELT PROCESSABILITY HEAT RESISTANCE GENERAL ELECTRIC COMPANY 2002-08-13 US disclosed
US-6388046-B1 MIXTURE CONTAINING THERMOPLASTIC RESIN GENERAL ELECTRIC COMPANY 2002-05-14 US disclosed
US-20020019466-A1 Method to prepare phosphoramides, and resin compositions containing them SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2002-02-14 US disclosed
EP-1144498-A1 FLAME RETARDANT POLYMER BLENDS, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2001-10-17 EP disclosed
EP-1131378-A1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2001-09-12 EP disclosed
EP-1115786-A1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2001-07-18 EP disclosed
US-6228912-B1 Flame retardant resin compositions containing phosphoramides and method for making GENERAL ELECTRIC COMPANY 2001-05-08 US disclosed
US-6221939-B1 THERMOPLASTIC RESIN BLEND GENERAL ELECTRIC COMPANY 2001-04-24 US disclosed
US-6204313-B1 AT LEAST ONE POLYESTERCARBONATE, AT LEAST ONE ADDITION POLYMER SUCH AS A STYRENE-ACRYLONITRILE OR ABS COPOLYMER, AND AT LEAST ONE PHOSPHORYL FLAME RETARDANT HAVE SUPERIOR HIGH TEMPERATURE STABILITY PROPERTIES GENERAL ELECTRIC COMPANY 2001-03-20 US disclosed
US-6174942-B1 COMPRISING BLEND OF POLYCARBONATE, ADDITION POLYMER AND PHOSPHORYL COMPOUND; FLAME RETARDANCE; DUCTILITY GENERAL ELECTRIC COMPANY 2001-01-16 US disclosed
WO-2000012613-A9 FLAME RETARDANT POLYMER BLENDS, AND METHOD FOR MAKING GEN ELECTRIC (US) 2000-08-17 WO disclosed
WO-2000012612-A1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2000-03-09 WO disclosed
WO-2000012613-A1 FLAME RETARDANT POLYMER BLENDS, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2000-03-09 WO disclosed
WO-2000012611-A1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2000-03-09 WO disclosed
WO-2000012609-A1 FLAME RETARDANT POLYMER BLENDS, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2000-03-09 WO disclosed
WO-2000012614-A1 FLAME RETARDANT RESIN COMPOSITIONS CONTAINING PHOSPHORAMIDES, AND METHOD FOR MAKING GENERAL ELECTRIC COMPANY (US) 2000-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019466-A1 Method to prepare phosphoramides, and resin compositions containing them PPA1, PHOSPHO1, PFAS MAPT 1823/4885CD44 3404/4885CYP3A4 4686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.