SCHEMBL5546431

SCHEMBL5546431

CCNc1c(NC(C)C)cccc1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.48
PKM P14618 1/20 0.48
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CLCN2 P51788 2/20 0.47
PIK3CA P42336 1/20 0.42
FABP4 P15090 1/20 0.42
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 3/20 0.39
AGTR1 P30556 1/20 0.39
RAB9A P51151 1/20 0.39
CXCR2 P25025 3/20 0.39
POLB P06746 2/20 0.38
ABCC1 P33527 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
AKR1B10 O60218 1/20 0.38
TRPA1 O75762 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236192 0.83 CLCN2 (0.50) MAPTPKMMAPK1SMN1; SMN2CLCN2
SCHEMBL28476762 0.82 MAPT (0.55) MAPTPKMMAPK1SMN1; SMN2CLCN2
SCHEMBL1899962 0.77 KMT2A (0.54) MAPTPKMCLCN2FABP4ALDH1A1
SCHEMBL6236190 0.76 CLCN2 (0.50) MAPTPKMMAPK1SMN1; SMN2CLCN2
SCHEMBL13073786 0.76 POLB (0.56) MAPTPKMMAPK1SMN1; SMN2CLCN2
SCHEMBL2413633 0.74 TSHR (0.52) MAPTMAPK1SMN1; SMN2CLCN2FABP4
SCHEMBL184136 0.73 ALDH1A1 (0.62) SMN1; SMN2CLCN2FABP4ALDH1A1HPGD
SCHEMBL16181442 0.72 FABP4 (0.50) MAPTCLCN2FABP4ALDH1A1HPGD
SCHEMBL21722620 0.72 KDM4E (0.48) MAPTMAPK1SMN1; SMN2ALDH1A1HPGD
SCHEMBL13073788 0.72 NPC1 (0.53) MAPTSMN1; SMN2CLCN2FABP4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651641-B1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LTD (GB) 2007-05-23 EP disclosed