SCHEMBL5546833

SCHEMBL5546833

O=C(NC1N=CC2=CN(S(=O)(=O)c3ccc(Cl)cc3)CCC2=N1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 1/20 0.42
FLT4 P35916 1/20 0.42
KDR P35968 1/20 0.42
CYP3A4 P08684 1/20 0.37
UTS2R Q9UKP6 1/20 0.36
MAPT P10636 2/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CHRNA7 P36544 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
NPC1 O15118 1/20 0.35
PGR P06401 1/20 0.35
CNR2 P34972 1/20 0.35
HTT P42858 1/20 0.35
PTPN1 P18031 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5546196 0.89 TRPV1 (0.38) UTS2R
SCHEMBL5540365 0.80 KMT2A (0.36) FLT1FLT4KDRMAPTCHRNA7
SCHEMBL5548485 0.78 KMT2A (0.37) MAPTMEN1KMT2A
SCHEMBL5546835 0.73 FLT1 (0.44) FLT1FLT4KDRCYP3A4MAPT
SCHEMBL5540977 0.72 DRD4 (0.46) MEN1KMT2ANPC1
SCHEMBL5540282 0.69 MCHR1 (0.42) CHRNA7ALDH1A1NPC1
SCHEMBL5545012 0.64 CCR3 (0.41) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL5546201 0.63 ABL1 (0.40) MEN1KMT2AHTT
SCHEMBL5546606 0.61 OPRK1 (0.35) MAPTMEN1KMT2AALDH1A1NPC1
SCHEMBL5540386 0.61 LMNA (0.34) MAPTMEN1KMT2AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed