SCHEMBL5540977

SCHEMBL5540977

O=C(NC1N=CC2=CN(C(=O)c3ccc4ccccc4c3)CCC2=N1)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 6/20 0.46
MCHR1 Q99705 1/20 0.45
SLC6A12 P48065 1/20 0.39
SLC6A13 Q9NSD5 1/20 0.39
HTR1A P08908 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CCR1 P32246 1/20 0.38
MGLL Q99685 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5544991 0.79 DRD4 (0.39) DRD4MEN1NPC1RAB9AKMT2A
SCHEMBL5540365 0.75 KMT2A (0.36) DRD4MCHR1MEN1NPC1RAB9A
SCHEMBL5545011 0.74 NPC1 (0.41) NPC1RAB9AKMT2A
SCHEMBL5544982 0.74 HPGDS (0.42) MCHR1MGLL
SCHEMBL5548485 0.73 KMT2A (0.37) MEN1RAB9AKMT2ACCR1MGLL
SCHEMBL5546833 0.72 FLT1 (0.42) MEN1NPC1KMT2A
SCHEMBL5546568 0.71 CHRM1 (0.38) MEN1KMT2A
SCHEMBL5546606 0.69 OPRK1 (0.35) DRD4MEN1NPC1RAB9AKMT2A
SCHEMBL5540386 0.69 LMNA (0.34) MEN1NPC1RAB9AKMT2ATDP1
SCHEMBL5544998 0.69 SIGMAR1 (0.41) DRD4MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed