SCHEMBL5546867

SCHEMBL5546867

COCCOCC(=O)N1C=C2C=NC(NC(=O)c3ccc(Cl)cc3)N=C2CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ACKR3 P25106 1/20 0.33
CXCR6 O00574 2/20 0.33
IDO1 P14902 1/20 0.33
CHRNA7 P36544 3/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
MMP2 P08253 1/20 0.32
EPHX2 P34913 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
NAMPT P43490 2/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5546932 0.80 TDP1 (0.36) MEN1KMT2ACHRNA7CHRNB2CHRNA4
SCHEMBL5546256 0.78 CHRNA7 (0.37) MEN1KMT2ACHRNA7CHRNB2CHRNA4
SCHEMBL5540977 0.75 DRD4 (0.46) MEN1KMT2ADRD4
SCHEMBL5545031 0.73 TP53 (0.38) MEN1KMT2ATSHR
SCHEMBL5540365 0.73 KMT2A (0.36) MEN1KMT2ACHRNA7HTR3EHTR3B
SCHEMBL5546870 0.73 NAMPT (0.34) KMT2AACKR3IDO1EPHX2NAMPT
SCHEMBL5546606 0.72 OPRK1 (0.35) MEN1KMT2ADRD4
SCHEMBL5540386 0.72 LMNA (0.34) MEN1KMT2AEPHX2
SCHEMBL5544998 0.70 SIGMAR1 (0.41) DRD2DRD4SLC6A5
SCHEMBL5548485 0.68 KMT2A (0.37) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed