SCHEMBL5546872

SCHEMBL5546872

O=C(NC1N=CC2=CN(S(=O)(=O)c3ccccc3C(F)(F)F)CCC2=N1)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.37
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
MEN1 O00255 2/20 0.35
KCNH2 Q12809 2/20 0.35
RAB9A P51151 1/20 0.34
MAPT P10636 2/20 0.34
CNR1 P21554 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
DCTPP1 Q9H773 1/20 0.34
POLB P06746 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALKBH2 Q6NS38 1/20 0.33
ALKBH3 Q96Q83 1/20 0.33
FTO Q9C0B1 1/20 0.33
BCAT1 P54687 2/20 0.33
HCRTR1 O43613 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548485 0.93 KMT2A (0.37) KMT2AITGB1ITGA4MEN1RAB9A
SCHEMBL5546875 0.75 MAPT (0.38) KMT2AITGB1ITGA4MEN1KCNH2
SCHEMBL5546833 0.74 FLT1 (0.42) KMT2AMEN1MAPTALDH1A1HTT
SCHEMBL5540365 0.71 KMT2A (0.36) KMT2AMEN1RAB9AMAPTALDH1A1
SCHEMBL5545012 0.69 CCR3 (0.41) KMT2AMEN1RAB9AMAPTPOLB
SCHEMBL5540282 0.69 MCHR1 (0.42) RAB9APOLBALDH1A1LMNA
SCHEMBL5540977 0.67 DRD4 (0.46) KMT2AMEN1RAB9A
SCHEMBL5545030 0.67 CYP2C9 (0.36) KCNH2HCRTR1LMNA
SCHEMBL5548490 0.67 MAPT (0.39) KMT2AMEN1RAB9AMAPTCNR1
SCHEMBL5544998 0.66 SIGMAR1 (0.41) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed