SCHEMBL5548598

SCHEMBL5548598

COc1ccc2ncc(F)c(N3CCN(CC(NC(=O)O)C(C)(C)C)CC3)c2n1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.39
SLC2A1 P11166 5/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2945463 0.81 KCNH2 (0.44) KCNH2SLC2A1KDM4EALDH1A1CYP1A2
SCHEMBL13238463 0.77 DRD2 (0.52) KCNH2KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL2952599 0.76 KCNH2 (0.42) KCNH2SLC2A1
SCHEMBL17844920 0.76 KCNH2 (0.48) KCNH2SLC2A1
SCHEMBL5548608 0.74 CYP8B1 (0.37) KCNH2SLC2A1
SCHEMBL17861460 0.72 CKS1B (0.48) KCNH2SLC2A1
SCHEMBL1224674 0.71 CHRNB2 (0.45) KCNH2ALDH1A1CYP1A2HSD17B10
SCHEMBL3632714 0.70 MAPT (0.42) KDM4EALDH1A1HSD17B10
SCHEMBL5260306 0.70 KCNH2 (0.51) KCNH2SLC2A1
SCHEMBL1222889 0.70 DPP4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1846411-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-10-24 EP disclosed
WO-2006081289-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2006-08-03 WO disclosed