SCHEMBL5548899

SCHEMBL5548899

CC(O)CNc1nc(C(C)(C)C)cn2c(=O)[nH]nc12

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.32
GSK3A P49840 12/20 0.32
ADORA1 P30542 2/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5550109 0.85 CASP1 (0.33) ADORA1
SCHEMBL5549142 0.85 GSK3B (0.35) GSK3BGSK3AADORA1
SCHEMBL3529268 0.83 ADORA1 (0.37) GSK3BGSK3AADORA1
SCHEMBL5545643 0.83 GSK3B (0.34) GSK3BGSK3AADORA1
SCHEMBL5549383 0.82 MAPT (0.40) ADORA3
SCHEMBL5548540 0.81 PDE5A (0.32) GSK3BGSK3A
SCHEMBL3522851 0.81 CXCR2 (0.35)
SCHEMBL5545590 0.81 GSK3B (0.35) GSK3BGSK3AADORA1
SCHEMBL3521775 0.81 GSK3B (0.36) GSK3BGSK3AADORA1
SCHEMBL5550132 0.79 ILK (0.35) GSK3BGSK3AADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed