SCHEMBL5550706

SCHEMBL5550706

Fc1ccc(NNC2CCCC2)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
TRPA1 O75762 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 2/20 0.45
MAPT P10636 2/20 0.45
HTT P42858 1/20 0.45
RAPGEF4 Q8WZA2 1/20 0.44
PLA2G1B P04054 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
NR1I2 O75469 1/20 0.43
AHR P35869 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15677756 0.77 RAB9A (0.53) ALDH1A1KMT2AMEN1SMN1; SMN2NPSR1
SCHEMBL5547469 0.76 LMNA (0.60) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL31453688 0.75 KMT2A (0.59) ALDH1A1KMT2AMEN1TRPA1NPSR1
SCHEMBL9008342 0.75 KMT2A (0.59) ALDH1A1KMT2AMEN1TRPA1NPSR1
SCHEMBL5550812 0.75 LMNA (0.62) ALDH1A1KMT2AMEN1MAPTCYP1A2
SCHEMBL25385990 0.73 PLA2G1B (0.57) ALDH1A1KMT2AMEN1NPSR1MAPT
SCHEMBL12218448 0.73 MEN1 (0.86) ALDH1A1KMT2AMEN1SMN1; SMN2HTT
SCHEMBL5550113 0.72 NPC1 (0.55) ALDH1A1KMT2AMEN1TRPA1SMN1; SMN2
SCHEMBL1241022 0.72 SOS1 (0.54) ALDH1A1KMT2AMEN1TRPA1SMN1; SMN2
SCHEMBL14465084 0.71 MEN1 (0.89) ALDH1A1KMT2AMEN1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002000649-A9 SUBSTITUTED QUINAZOLINE DERIVATIVES AND THEIR USE AS INHIBITORS ASTRAZENECA AB (SE) 2007-09-20 WO disclosed
EP-1299381-A1 SUBSTITUTED QUINAZOLINE DERIVATIVES AND THEIR USE AS INHIBITORS AstraZeneca AB (SE) 2003-04-09 EP disclosed
WO-2002000649-A1 SUBSTITUTED QUINAZOLINE DERIVATIVES AND THEIR USE AS INHIBITORS ASTRAZENECA AB (SE) 2002-01-03 WO disclosed