SCHEMBL5551290

SCHEMBL5551290

O=C(CN1CCC(Br)C1=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CYP2C19 P33261 3/20 0.43
FKBP1A P62942 3/20 0.43
CYP2C9 P11712 2/20 0.42
CYP1A2 P05177 1/20 0.42
CDC25B P30305 1/20 0.42
CYP3A4 P08684 1/20 0.41
GLA P06280 1/20 0.41
ACE P12821 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5551252 0.92 ALDH1A1 (0.43) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL17949283 0.84 SMN1; SMN2 (0.46) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL8082401 0.80 SMN1; SMN2 (0.44) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL15368459 0.80 PER2 (0.45) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL4985094 0.79 CASP3 (0.46) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
Hydrochloric Acid SCHEMBL8082397 0.79 SMN1; SMN2 (0.43) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
Hydrochloric Acid SCHEMBL8082404 0.79 SMN1; SMN2 (0.43) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL4985086 0.79 CASP3 (0.46) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
SCHEMBL5038822 0.78 GLA (0.42) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1
Hydrochloric Acid SCHEMBL10795974 0.78 CASP3 (0.46) ALDH1A1MAPK1L3MBTL1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1301750-C Conjugates of macrocyclic metal complexes with biomolucules and utilization thereof for producing agents for use in NMR diagnosis and radiodiagnosis and radiotherapy SCHERING AG (DE) 2007-02-28 CN disclosed
US-20070014725-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy SCHERING AG (DE) 2007-01-18 US disclosed
US-7164016-B2 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2007-01-16 US disclosed
US-20070009442-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2007-01-11 US disclosed
CN-1541114-A Conjugates of macrocyclic metal complexes with biomolucules and utilization thereof for producing agents for use in NMR diagnosis and radiodiagnosis and radiotherapy ���ֹɷݹ�˾ 2004-10-27 CN disclosed
CN-1533286-A Macrocyclic metal complexes and use thereof for production of conjugates with biomolecules ���ֹɷݹ�˾ 2004-09-29 CN disclosed
US-20030206865-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy SCHERING AG (DE) 2003-11-06 US disclosed
US-20030108486-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2003-06-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030108486-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules CA13, MPI, CA14 ALDH1A1 3392/4885MAPK1 3917/4885L3MBTL1 3120/4885
US-20070014725-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy CA13, CA14, CA12 ALDH1A1 2758/4885MAPK1 3745/4885L3MBTL1 3119/4885
US-20030206865-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy CA13, CA14, CA12 ALDH1A1 2758/4885MAPK1 3745/4885L3MBTL1 3119/4885
US-20070009442-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules CA13, MPI, CA14 ALDH1A1 3392/4885MAPK1 3917/4885L3MBTL1 3120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.