SCHEMBL5553751

SCHEMBL5553751

N[C@@H]1CC[C@@H](c2cccc(F)c2F)CN(C(=O)O)C1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 11/20 0.41
HPGD P15428 1/20 0.38
NOTUM Q6P988 1/20 0.37
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12812342 0.86 HCRTR2 (0.42) CALCRLHPGDNOTUMHCRTR2
SCHEMBL1434918 0.82 SMN1; SMN2 (0.46)
SCHEMBL5552182 0.82 SMN1; SMN2 (0.46)
SCHEMBL30663898 0.77 RBP4 (0.47) CALCRLHPGDNOTUMHCRTR2
SCHEMBL12812347 0.77 HCRTR2 (0.41) CALCRLHCRTR2
SCHEMBL1434919 0.77 DRD2 (0.41) CALCRL
SCHEMBL12812343 0.76 NAMPT (0.41) CALCRLHCRTR2
SCHEMBL12812349 0.75 HPGD (0.48) CALCRLHPGD
SCHEMBL5553762 0.74 CA1 (0.43) CALCRLHCRTR2
SCHEMBL12812368 0.73 HCRTR2 (0.41) CALCRLHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804919-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047196-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed