SCHEMBL5560933

SCHEMBL5560933

CCc1c(CO)nn(C(C)C)c1Oc1ccc(C#N)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PGR P06401 9/20 0.39
HRH3 Q9Y5N1 3/20 0.36
LCK P06239 1/20 0.35
KDR P35968 1/20 0.35
TEK Q02763 1/20 0.35
KDM4E B2RXH2 1/20 0.35
SCN9A Q15858 6/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5561726 0.88 KCNH2 (0.40)
SCHEMBL5555674 0.86 EPAS1 (0.41) HRH3KDRSCN9A
SCHEMBL5560668 0.84 MAPT (0.37) HRH3KDM4E
SCHEMBL5561581 0.84 PGR (0.41) PGRHRH3KDM4E
SCHEMBL5562337 0.83 KCNH2 (0.45)
SCHEMBL5555878 0.72 EPAS1 (0.38) HRH3SCN9A
SCHEMBL14471297 0.70 PGR (0.41) PGRKDM4E
SCHEMBL5560889 0.69 KCNH2 (0.34)
SCHEMBL5560926 0.69 KCNH2 (0.47)
SCHEMBL5562173 0.69 EPAS1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed