Maleic Acid

Maleic Acid

SCHEMBL5556979

O=C(O)/C=C\C(=O)O.O=C(O)O.O=C(O)O

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.90
TP53 P04637 1/20 0.90
EGLN1 Q9GZT9 1/20 0.90
EGLN3 Q9H6Z9 1/20 0.90
HCAR2 Q8TDS4 4/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
GABRR1 P24046 2/20 0.44
GABRR2 P28476 2/20 0.44
BLM P54132 2/20 0.44
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
GABRR3 A8MPY1 1/20 0.44
APEX1 P27695 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7568616 1.00 TSHR (0.90) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL4838658 1.00 TSHR (0.90) TSHRTP53EGLN1EGLN3HCAR2
Maleic Acid SCHEMBL4838648 1.00 TSHR (0.90) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL8584098 0.95 TSHR (0.82) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL3254191 0.95 TSHR (0.82) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL2046433 0.95 TSHR (1.00) TSHRTP53EGLN1EGLN3HCAR2
Maleic Acid SCHEMBL2046430 0.95 TSHR (1.00) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL3998225 0.95
Maleic Acid SCHEMBL20487516 0.95 TSHR (1.00) TSHRTP53EGLN1EGLN3HCAR2
Fumaric Acid SCHEMBL6875 0.95 TSHR (1.00) TSHRTP53EGLN1EGLN3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1752526-A2 Solid detergent compositions The Procter and Gamble Company (US) 2007-02-14 EP disclosed
EP-1752527-A2 Solid detergent compositions THE PROCTER & GAMBLE COMPANY (US) 2007-02-14 EP disclosed
EP-1728851-A2 Solid detergent compositions The Procter & Gamble Company (US) 2006-12-06 EP disclosed
EP-1728850-A2 Solid detergent compositions The Procter and Gamble Company (US) 2006-12-06 EP disclosed
EP-1115835-B1 SOLID DETERGENT COMPOSITIONS PROCTER & GAMBLE (US) 2006-05-31 EP disclosed
EP-1124929-B1 BLEACH-CONTAINING DETERGENT COMPOSITION PROCTER & GAMBLE (US) 2005-07-27 EP disclosed
CN-1454252-A Detergent compositions comprising a maltogenic alpha-amylase enzyme PROCTER & GAMBLE (US) 2003-11-05 CN disclosed
US-6627597-B1 Granular form and in a nanoporous anhydrous state, a process for improving the water-solubility and controlled release characteristics of a detergent material, and a detergent composition are disclosed. THE PROCTER & GAMBLE COMPANY 2003-09-30 US disclosed
US-6555514-B1 For cold temperature laundering solutions THE PROCTER & GAMBLE COMPANY 2003-04-29 US disclosed
EP-1124937-B1 PROCESSES FOR MAKING GRANULAR DETERGENT COMPOSITION HAVING IMPROVED APPEARANCE AND SOLUBILITY PROCTER & GAMBLE (US) 2002-12-11 EP disclosed