SCHEMBL5557458

SCHEMBL5557458

Cc1cccc(C(=O)Nc2cc3ccccc3[nH]2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
KCNK3 O14649 5/20 0.54
KCNK9 Q9NPC2 4/20 0.54
KCNH2 Q12809 1/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.51
GRM5 P41594 1/20 0.51
FOXO1 Q12778 1/20 0.51
RXFP1 Q9HBX9 2/20 0.50
TP53 P04637 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
KDM4E B2RXH2 1/20 0.50
TSHR P16473 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
EGFR P00533 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433791 0.85 NPC1 (0.58) NPC1RAB9AKCNK3KCNK9SMN1; SMN2
SCHEMBL13801599 0.81 NPC1 (0.50) MEN1KMT2ANPC1RAB9APOLB
SCHEMBL4352826 0.77 TOP1 (0.55) NPC1RAB9ASMN1; SMN2KDM4EEGFR
SCHEMBL9269321 0.77 GRIK1 (0.56) NPC1RAB9ASMN1; SMN2KDM4EEGFR
SCHEMBL3569428 0.76 NPC1 (0.71) NPC1RAB9ASMN1; SMN2KDM4EEGFR
SCHEMBL8558926 0.76 RAB9A (0.81) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL4413986 0.76 MTNR1A (0.53) KMT2ANPC1RAB9APOLBSMN1; SMN2
SCHEMBL31487774 0.76 MTNR1A (0.53) KMT2ANPC1RAB9APOLBSMN1; SMN2
SCHEMBL10227495 0.75 PDGFRB (0.68) MEN1KMT2ANPC1RAB9ARXFP1
SCHEMBL22488995 0.75 FOXO1 (0.68) MEN1KMT2ANPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756112-A1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS Boehringer Ingelheim International GmbH (DE) 2007-02-28 EP disclosed
WO-2005111040-A1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed