SCHEMBL5558076

SCHEMBL5558076

Cc1cc(N)c2cccc(NC(=O)c3ccc(CNc4cc(C)[n+](C)c(N)n4)cc3)c2n1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 0.52
HDAC6 Q9UBN7 2/20 0.42
HDAC2 Q92769 3/20 0.41
HDAC3 O15379 2/20 0.41
NCOR2 Q9Y618 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX12 P18054 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CD38 P28907 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5558113 0.84 CD38 (0.44) HDAC6CD38
SCHEMBL5558052 0.82 DNMT1 (0.47) MEN1ALDH1A1ALOX12RAB9AKMT2A
SCHEMBL3233220 0.81 MMP9 (0.51) HDAC6MEN1KMT2A
SCHEMBL3243944 0.80 MMP9 (0.46) HDAC6MEN1KMT2A
SCHEMBL1062263 0.72 HDAC1 (0.76) HDAC1HDAC6HDAC2HDAC3NCOR2
SCHEMBL5559910 0.72 DNMT1 (0.45) HDAC6
SCHEMBL5558936 0.71 DNMT1 (0.47) HDAC6
SCHEMBL5558101 0.70 CD38 (0.48) MEN1KMT2ACD38
SCHEMBL1064771 0.69 HDAC1 (1.00) HDAC1HDAC6HDAC2HDAC3NCOR2
SCHEMBL3245888 0.69 MMP9 (0.49) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1509516-B1 INHIBITORS OF THE GPIB -VWF INTERACTION, THEIR PREPARATION AND USE SANOFI AVENTIS DEUTSCHLAND (DE) 2007-01-31 EP claimed