SCHEMBL5560484

SCHEMBL5560484

CCC(C)OC(=O)C(C)c1c(C)n(C(=O)c2ccc(Cl)c(Cl)c2)c2ccc(O)c(F)c12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
PTGS2 P35354 8/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
MGLL Q99685 1/20 0.33
ABCB11 O95342 1/20 0.32
AKR1C3 P42330 2/20 0.32
AKR1C2 P52895 2/20 0.32
SLC6A2 P23975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822267 0.94 PTGS2 (0.33) PTGS2MGLLAKR1C3AKR1C2
SCHEMBL5800263 0.91 TSHR (0.39) TSHRPTGS2ABCB11AKR1C3AKR1C2
SCHEMBL5801225 0.91 PTGS2 (0.36) TSHRPTGS2ABCB11AKR1C3AKR1C2
SCHEMBL5800266 0.91 TSHR (0.39) TSHRPTGS2ABCB11AKR1C3AKR1C2
SCHEMBL5801230 0.91 PTGS2 (0.36) TSHRPTGS2ABCB11AKR1C3AKR1C2
SCHEMBL5797099 0.90 PTGS2 (0.40) PTGS2AKR1C3AKR1C2
SCHEMBL5798904 0.89 TSHR (0.35) TSHRPTGS2SLC6A4SLC6A3MGLL
SCHEMBL5559072 0.89 ELANE (0.37) PTGS2MGLL
SCHEMBL6423511 0.89 ELANE (0.37) PTGS2MGLL
SCHEMBL5800364 0.88 PTGS2 (0.38) TSHRPTGS2ABCB11AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed