SCHEMBL5560554

SCHEMBL5560554

CC[C@H](C)c1c(O)ccc2c1c(OC(C)=O)c(C)n2C(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.40
PPARG P37231 11/20 0.39
PPARA Q07869 5/20 0.39
EPHX2 P34913 1/20 0.36
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
PTGS2 P35354 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5559328 1.00 HRH3 (0.40) HRH3PPARGPPARAEPHX2AKR1C3
SCHEMBL5558544 0.88 PTGS2 (0.34) PPARGPPARAAKR1C3AKR1C2PTGS2
SCHEMBL5560462 0.88 PTGS2 (0.34) PPARGPPARAAKR1C3AKR1C2PTGS2
SCHEMBL5798576 0.86 PTGS2 (0.41) PPARGAKR1C3AKR1C2PTGS2
SCHEMBL5554254 0.86 PTGS2 (0.34) AKR1C3AKR1C2PTGS2
SCHEMBL5554445 0.84 PPARG (0.37) HRH3PPARGPPARAAKR1C3AKR1C2
SCHEMBL5560446 0.82 HRH3 (0.39) HRH3PPARGPPARAEPHX2TRPV1
SCHEMBL5560599 0.81 LMNA (0.39) AKR1C3AKR1C2
SCHEMBL5560527 0.81 PTGS2 (0.33) AKR1C3AKR1C2PTGS2
SCHEMBL5559277 0.78 SCN9A (0.37) HRH3PPARGPPARATRPV1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed