SCHEMBL5564013

SCHEMBL5564013

CC1(C)C(=O)N(CCOC2CC2)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ACHE P22303 1/20 0.37
PNMT P11086 4/20 0.37
ADRA2A P08913 3/20 0.37
ADRA2B P18089 2/20 0.37
ADRA2C P18825 2/20 0.37
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
CASP1 P29466 1/20 0.34
CASP3 P42574 1/20 0.34
CASP4 P49662 1/20 0.34
CASP7 P55210 1/20 0.34
CASP9 P55211 1/20 0.34
CASP6 P55212 1/20 0.34
AKR1B1 P15121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5555976 0.82 ACHE (0.52) HTTALDH1A1SMN1; SMN2ACHEPNMT
SCHEMBL2487541 0.81 TDP1 (0.49) HTTALDH1A1SMN1; SMN2GAAL3MBTL1
SCHEMBL5562474 0.78 ESPL1 (0.40) HTTSMN1; SMN2ACHEADRA2AL3MBTL1
SCHEMBL4507178 0.78 CYP1A2 (0.46) ALDH1A1L3MBTL1LMNAMAPTCASP1
SCHEMBL2487312 0.77 BACE1 (0.33) LMNA
SCHEMBL5561087 0.76 F2RL3 (0.43) ALDH1A1L3MBTL1MAPTCASP1CASP3
SCHEMBL15577345 0.76 CYP19A1 (0.33) LMNA
SCHEMBL15577409 0.76 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2MAPT
SCHEMBL5555736 0.75 ESPL1 (0.38) HTTALDH1A1SMN1; SMN2PNMTADRA2A
SCHEMBL26621510 0.75 L3MBTL1 (0.38) HTTALDH1A1SMN1; SMN2ACHEL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756112-A1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS Boehringer Ingelheim International GmbH (DE) 2007-02-28 EP disclosed
WO-2005111040-A1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed