SCHEMBL5566700

SCHEMBL5566700

Cc1ccc(-c2nc3ccccn3c2CC=O)cc1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.65
NPC1 O15118 4/20 0.65
RAB9A P51151 4/20 0.65
MAPK1 P28482 1/20 0.52
KDM4E B2RXH2 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
POLB P06746 1/20 0.51
HTT P42858 1/20 0.51
KCNK3 O14649 4/20 0.51
KCNK9 Q9NPC2 4/20 0.51
MAPT P10636 1/20 0.48
GABRA1 P14867 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRB2 P47870 1/20 0.47
ADORA1 P30542 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13341898 0.89 NPC1 (0.54) ALDH1A1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL13368337 0.86 KDM4E (0.64) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL2932378 0.83 GABRA1 (0.61) ALDH1A1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL18978250 0.83 NPC1 (0.59) ALDH1A1NPC1RAB9AMAPK1KDM4E
SCHEMBL9999613 0.82 DPP4 (0.66) ALDH1A1NPC1RAB9AMAPK1KDM4E
SCHEMBL1691474 0.82 ALDH1A1 (0.58) ALDH1A1NPC1RAB9AMAPK1KDM4E
Hydrochloric Acid SCHEMBL1430695 0.81 NPC1 (0.57) ALDH1A1NPC1RAB9AMAPK1KDM4E
SCHEMBL1779622 0.80 KMT2A (0.50) ALDH1A1NPC1RAB9AMAPK1KDM4E
SCHEMBL28372805 0.80 NPC1 (0.56) ALDH1A1NPC1RAB9AMAPK1KDM4E
SCHEMBL22635913 0.79 KCNK3 (0.66) ALDH1A1NPC1RAB9AKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120122874-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR TREATING DEPRESSION Sunovion Inc. (US) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122874-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR TREATING DEPRESSION HTR2A, HTR5A, HTR2C ALDH1A1 421/4885NPC1 2142/4885RAB9A 779/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.