SCHEMBL5568496

SCHEMBL5568496

[c]1nnnc2cccc(-c3cnc4ccccc4n3)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.43
RAB9A P51151 8/20 0.43
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK10 P53779 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
ALOX12 P18054 1/20 0.40
ATM Q13315 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
BCHE P06276 1/20 0.40
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADORA3 P0DMS8 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065135 0.73 HTR2C (0.34)
SCHEMBL27775278 0.71 NPC1 (0.53) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL2243516 0.69 KDM4E (0.52) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL3076524 0.69 NPC1 (0.63) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL29942654 0.69 NPC1 (0.63) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL29614829 0.69 NPC1 (0.63) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL29966674 0.69 NPC1 (0.63) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL2076567 0.68 HSP90AA1 (0.57) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL9453979 0.67 ALDH1A1 (0.66) NPC1RAB9AKMT2AALDH1A1MAPK10
SCHEMBL4232322 0.67 NPC1 (0.53) NPC1RAB9AKMT2AALDH1A1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2007-05-02 EP disclosed
WO-2006020049-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2006-02-23 WO disclosed