SCHEMBL5569734

SCHEMBL5569734

Cc1ccc(S(=O)(=O)N(CC(=O)N[C@@H](Cc2ccccc2)C(=O)O)C(C)c2cccs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.44
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
ALDH1A1 P00352 2/20 0.44
ITGB1 P05556 2/20 0.43
ITGA4 P13612 2/20 0.43
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
POLB P06746 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GAA P10253 1/20 0.41
MMP9 P14780 1/20 0.41
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
CA2 P00918 2/20 0.40
ACE P12821 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28745281 0.84 ALDH1A1 (0.39) ALDH1A1ITGB1ITGA4HTTSMN1; SMN2
SCHEMBL7365612 0.81 DAGLA (0.48) POLBTDP1MMP9TP53
SCHEMBL5569737 0.79 CA12 (0.50) CA1CA12CA9ALDH1A1TP53
SCHEMBL5572753 0.79 SMN1; SMN2 (0.55) CA1CA12CA9ALDH1A1ITGB1
SCHEMBL5573330 0.77 MEN1 (0.58) CA1CA12CA9ALDH1A1ITGB1
SCHEMBL5574133 0.77 THRB (0.61) CA1CA12CA9ALDH1A1HTT
SCHEMBL5570733 0.75 ALDH1A1 (0.60) CA1CA12CA9ALDH1A1SMN1; SMN2
SCHEMBL5496683 0.72 LMNA (0.61) ALDH1A1HTTSMN1; SMN2POLBTDP1
SCHEMBL5496678 0.72 LMNA (0.61) ALDH1A1HTTSMN1; SMN2POLBTDP1
SCHEMBL5569686 0.71 MEN1 (0.51) ALDH1A1TP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7166580-B2 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2007-01-23 US claimed
US-20030166575-A1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 BIOGEN MA INC. 2003-09-04 US claimed
EP-1001973-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006433-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-7166580-B2 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2007-01-23 US disclosed
US-20030166575-A1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 BIOGEN MA INC. 2003-09-04 US disclosed
US-6559127-B1 Intercellular adhesion mediated by VLA-4 and other cell surface receptors is associated with a number of inflammatory responses ATHENA NEUROSCIENCES, INC. 2003-05-06 US disclosed
EP-1001973-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP disclosed
WO-1999006433-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030166575-A1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 VCAM1, ICAM1, CD4 CA1 916/4885CA12 2790/4885CA9 2934/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.