SCHEMBL5569860

SCHEMBL5569860

CC1Cc2ccc(CC(N)=O)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TBXA2R P21731 5/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530910 0.85 KDM4E (0.46) CA2KDM4EALDH1A1TBXA2RLMNA
SCHEMBL11531134 0.81 ALDH1A1 (0.49) ALDH1A1TBXA2R
SCHEMBL15338335 0.77 HTR2A (0.44)
SCHEMBL16526945 0.75 MAPK8 (0.54) CA2ALDH1A1LMNA
SCHEMBL11862393 0.75 ACHE (0.58) CA2
SCHEMBL658778 0.74 MAPK8 (0.55) CA2ALDH1A1LMNA
SCHEMBL31339549 0.74 MAPK8 (0.55) CA2ALDH1A1LMNA
SCHEMBL3800131 0.72 CA2 (0.46) CA2KDM4EALDH1A1LMNAPOLB
SCHEMBL24997114 0.72 CTSD (0.42) SLC6A2SLC6A4
SCHEMBL9472297 0.71 CA2 (0.47) CA2KDM4EALDH1A1TBXA2RLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866292-A1 TRICYCLIC 1,2,4-TRIAZINE OXIDES AND COMPOSITIONS THEREFROM FOR THERAPEUTIC USE IN CANCER TREATMENTS Auckland Uniservices Limited (NZ) 2007-12-19 EP disclosed
WO-2006104406-A1 TRICYCLIC 1,2,4-TRIAZINE OXIDES AND COMPOSITIONS THEREFROM FOR THERAPEUTIC USE IN CANCER TREATMENTS AUCKLAND UNISERVICES LIMITED (NZ) 2006-10-05 WO disclosed