SCHEMBL5571722

SCHEMBL5571722

CS(=O)(=O)C(CO)(NS(=O)(=O)c1cccc(C(N)=O)c1)S(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
F2 P00734 6/20 0.42
PRSS1 P07477 3/20 0.42
PRSS2 P07478 3/20 0.42
PRSS3 P35030 3/20 0.42
GAA P10253 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
LMNA P02545 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032668 0.84 ALDH1A1 (0.50) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL5032686 0.84 CYP2C19 (0.45) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL5571728 0.82 F2 (0.48) F2PRSS1PRSS2PRSS3CA1
SCHEMBL5041352 0.80 LMNA (0.61) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL5566210 0.76 CA1 (0.56) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL28208130 0.76 ADAMTS4 (0.50) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL2854385 0.75 LMNA (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2850555 0.75 LMNA (0.53) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL5041380 0.74 CYP2C19 (0.49) CYP2C19HDAC3HDAC4HDAC1HDAC7
SCHEMBL5034887 0.73 CYP2C19 (0.76) CYP2C19HDAC2HDAC8HDAC6PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-A1 PYRRAZOLO-PYRIMIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005123738-A1 PYRRAZOLO-PYRIMIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2005-12-29 WO disclosed