SCHEMBL5577609

SCHEMBL5577609

COc1ccc(CN2CCCN(c3ncc(CNC(=O)c4cccc(Cl)c4C)s3)CC2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.46
TP53 P04637 2/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
KDM4E B2RXH2 3/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
THRB P10828 1/20 0.41
POLB P06746 1/20 0.41
ABCB1 P08183 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C8 P10632 2/20 0.41
CYP2C19 P33261 2/20 0.41
LMNA P02545 2/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5577386 0.97 ALDH1A1 (0.44) ALDH1A1TP53KMT2AMEN1KDM4E
SCHEMBL5577678 0.88 MT-CO2 (0.44) ALDH1A1TP53KMT2AMEN1KDM4E
SCHEMBL5577473 0.86 ALDH1A1 (0.51) ALDH1A1TP53POLBLMNAHPGD
SCHEMBL5577758 0.85 LMNA (0.41) ALDH1A1TP53THRBLMNAHPGD
SCHEMBL5577710 0.85 ALDH1A1 (0.40) ALDH1A1KMT2AMEN1KDM4ETHRB
SCHEMBL5577861 0.84 ALDH1A1 (0.49) ALDH1A1KMT2AMEN1KDM4EALOX15
SCHEMBL5577474 0.84 MT-CO2 (0.46) ALDH1A1TP53LMNASMN1; SMN2
SCHEMBL5577827 0.84 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1KDM4EALOX15
SCHEMBL5577633 0.84 JAK1 (0.43) ALDH1A1KMT2AMEN1KDM4EABCB1
SCHEMBL5577522 0.84 LMNA (0.45) ALDH1A1KMT2AMEN1KDM4EALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-02-22 US disclosed
EP-1616862-A1 NITROGENOUS HETEROCYCLIC COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-01-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof HLA-DRB1, MIF, HLA-C ALDH1A1 1147/4885TP53 397/4885KMT2A 3527/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.