SCHEMBL5582056

SCHEMBL5582056

C[Si](C)(C)CC(NC(=O)c1cccc(I)c1)C(=O)N(C#N)C1CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 5/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
CTSL P07711 9/20 0.35
CTSS P25774 5/20 0.35
CTSK P43235 4/20 0.35
GRM5 P41594 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MYC P01106 1/20 0.35
MAX P61244 1/20 0.35
TP53BP1 Q12888 1/20 0.34
CTSV O60911 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MTOR P42345 1/20 0.34
CTSF Q9UBX1 1/20 0.34
PRKD1 Q15139 2/20 0.34
PRKD3 O94806 1/20 0.34
PRKD2 Q9BZL6 1/20 0.34
SLC6A2 P23975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5581287 0.84 CTSS (0.48) CTSBCTSLCTSSCTSKCTSV
SCHEMBL5582057 0.80 TP53BP1 (0.39) HDAC1HDAC2CTSLCTSSGRM5
SCHEMBL5516526 0.77 HDAC1 (0.45) HDAC1HDAC2GRM5MYCMAX
SCHEMBL5516521 0.77 HDAC1 (0.45) HDAC1HDAC2GRM5MYCMAX
SCHEMBL5520013 0.75 CTSL (0.57) CTSBCTSLCTSSCTSK
SCHEMBL5520008 0.75 CTSL (0.57) CTSBCTSLCTSSCTSK
SCHEMBL5514133 0.73 HDAC1 (0.44) HDAC1HDAC2GRM5MYCMAX
SCHEMBL5514129 0.73 HDAC1 (0.44) HDAC1HDAC2GRM5MYCMAX
SCHEMBL5531439 0.71 CTSL (0.50) CTSBCTSLCTSSCTSK
SCHEMBL6048161 0.70 CTSS (0.46) CTSBCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007519744-A 2007-07-19 JP claimed
EP-1716158-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Schering Aktiengesellschaft (DE) 2006-11-02 EP claimed
WO-2005074904-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2005-08-18 WO claimed
EP-1716158-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Schering Aktiengesellschaft (DE) 2006-11-02 EP disclosed
WO-2005074904-A2 SILINANE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2005-08-18 WO disclosed