SCHEMBL5583491

SCHEMBL5583491

Clc1ccccc1-c1c(Cl)ccc2c1O[CH]C2

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDK2 Q15119 1/20 0.34
ADORA2A P29274 1/20 0.31
NOTUM Q6P988 1/20 0.31
AHR P35869 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958298 0.85 NPC1 (0.33) CYP2A6NPC1TP53HPGDRAB9A
SCHEMBL8251647 0.71 AXL (0.34) CYP2A6NPC1TP53HPGDRAB9A
SCHEMBL4609617 0.70 AQP1 (0.36) AHRGABRA1GABRG2GABRB3
SCHEMBL5586510 0.70 AQP1 (0.38) CYP2A6NPC1TP53HPGDRAB9A
SCHEMBL4596283 0.70 HTR1A (0.44) GABRA1GABRG2GABRB3
SCHEMBL4596281 0.70 GABRA1 (0.34) CYP2A6NPC1TP53HPGDRAB9A
SCHEMBL4230148 0.67 AQP1 (0.46) GABRA1GABRG2GABRB3DPP4
SCHEMBL4964386 0.67 AQP1 (0.42) PDK2GABRA1GABRG2GABRB3
SCHEMBL5583500 0.67 CSNK2A2 (0.34) NPC1HPGDRAB9ASMN1; SMN2DPP4
SCHEMBL4230244 0.67 AQP1 (0.42) CYP2A6PDK2GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed