SCHEMBL5583518

SCHEMBL5583518

CC1Cc2cc(Cl)cc(-c3ccc(F)c(F)c3)c2O1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
HTR1A P08908 4/20 0.37
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
CREBBP Q92793 1/20 0.35
BRD4 O60885 1/20 0.35
USP7 Q93009 1/20 0.35
AQP1 P29972 2/20 0.34
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597199 0.90 GRM2 (0.42) PARP1PTGS1PTGS2HTR1ACREBBP
SCHEMBL5583517 0.83 USP7 (0.37) PTGS1PTGS2PRKAB2PRKAG1PRKAA2
SCHEMBL4597185 0.83 MAOA (0.36) PARP1PTGS1PTGS2HTR1APRKAB2
SCHEMBL4596855 0.81 HTR2A (0.43) PARP1HTR1ACREBBPBRD4AQP1
SCHEMBL4596570 0.81 AQP1 (0.41) PARP1HTR1AAQP1GRM2
SCHEMBL4220019 0.80 PRKAB2 (0.58) PTGS1PTGS2PRKAB2PRKAG1PRKAA2
SCHEMBL4231239 0.80 AQP1 (0.58) PTGS1PTGS2PRKAB2PRKAG1PRKAA2
SCHEMBL4712018 0.80 AQP1 (0.40) PARP1HTR1AAQP1GRM2
SCHEMBL4231244 0.79 PRKAB2 (0.48) PTGS1PTGS2PRKAB2PRKAG1PRKAA2
SCHEMBL4963750 0.79 PARP1 (0.48) PARP1PTGS1PTGS2HTR1ABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed