SCHEMBL5591156

SCHEMBL5591156

CN1CCN(C2CCN(Cc3cccc(C(=O)NN(CC4CCCC4)c4nc(C#N)ncc4Br)c3)CC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.56
CTSK P43235 5/20 0.56
CTSL P07711 4/20 0.56
CTSB P07858 1/20 0.56
CXCR3 P49682 5/20 0.38
RORC P51449 1/20 0.37
WNT1 P04628 2/20 0.36
GSK3B P49841 2/20 0.36
DYRK1A Q13627 2/20 0.36
ACKR3 P25106 2/20 0.36
MBTD1 Q05BQ5 1/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5591406 0.94 CTSS (0.63) CTSSCTSKCTSLCTSBRORC
SCHEMBL5590944 0.92 CTSS (0.68) CTSSCTSKCTSLCTSBCXCR3
SCHEMBL8244996 0.90 CTSL (0.43) CTSSCTSKCTSLCTSBCXCR3
SCHEMBL3165237 0.90 CTSS (0.53) CTSSCTSKCTSLCTSBCXCR3
SCHEMBL3159740 0.89 CTSS (0.52) CTSSCTSKCTSLCTSBCXCR3
SCHEMBL5591180 0.89 CTSS (0.68) CTSSCTSKCTSLCTSBCXCR3
Trifluoroacetic Acid SCHEMBL5591334 0.87 CTSS (0.62) CTSSCTSKCTSLCTSBCXCR3
SCHEMBL5591423 0.85 CTSS (0.76) CTSSCTSKCTSLCTSBHDAC3
Trifluoroacetic Acid SCHEMBL3175934 0.85 CTSS (0.49) CTSSCTSKCTSLCTSBCXCR3
Trifluoroacetic Acid SCHEMBL3160111 0.85 CTSS (0.48) CTSSCTSKCTSLCTSBCXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed