SCHEMBL5591406

SCHEMBL5591406

CN1CCN(Cc2cccc(C(=O)NN(CC3CCCC3)c3nc(C#N)ncc3Br)c2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.63
CTSK P43235 5/20 0.63
CTSL P07711 4/20 0.63
CTSB P07858 1/20 0.63
RORC P51449 1/20 0.41
WNT1 P04628 3/20 0.40
GSK3B P49841 3/20 0.40
DYRK1A Q13627 3/20 0.40
HDAC3 O15379 4/20 0.39
HDAC4 P56524 4/20 0.39
HDAC1 Q13547 4/20 0.39
HDAC7 Q8WUI4 4/20 0.39
HDAC2 Q92769 4/20 0.39
HDAC10 Q969S8 4/20 0.39
HDAC11 Q96DB2 4/20 0.39
HDAC8 Q9BY41 4/20 0.39
HDAC6 Q9UBN7 4/20 0.39
HDAC9 Q9UKV0 4/20 0.39
HDAC5 Q9UQL6 4/20 0.39
CHRM3 P20309 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5591156 0.94 CTSS (0.56) CTSSCTSKCTSLCTSBRORC
SCHEMBL5591423 0.91 CTSS (0.76) CTSSCTSKCTSLCTSBHDAC3
SCHEMBL5591381 0.87 CTSL (0.60) CTSSCTSKCTSLCTSB
SCHEMBL5591471 0.87 CTSS (0.69) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL3165448 0.86 CTSS (0.52) CTSSCTSKCTSLCTSBRORC
SCHEMBL5591574 0.86 CTSS (0.63) CTSSCTSKCTSLCTSBGSK3B
SCHEMBL3174606 0.86 CTSS (0.55) CTSSCTSKCTSLCTSBRORC
Trifluoroacetic Acid SCHEMBL5591441 0.86 CTSS (0.69) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL3159651 0.86 CTSS (0.51) CTSSCTSKCTSLCTSBRORC
SCHEMBL3166071 0.85 CTSS (0.54) CTSSCTSKCTSLCTSBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed