SCHEMBL8244996

SCHEMBL8244996

CN1CCN(C2CCN(Cc3cccc(C(=O)NN(CC4CCCC4)c4nc(N)ncc4Br)c3)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
WNT1 P04628 2/20 0.38
GSK3B P49841 2/20 0.38
DYRK1A Q13627 2/20 0.38
MBTD1 Q05BQ5 1/20 0.37
L3MBTL3 Q96JM7 1/20 0.37
ACKR3 P25106 1/20 0.37
PDGFRB P09619 1/20 0.37
KDR P35968 1/20 0.37
HDAC3 O15379 3/20 0.36
HDAC4 P56524 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC7 Q8WUI4 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC10 Q969S8 3/20 0.36
HDAC11 Q96DB2 3/20 0.36
HDAC8 Q9BY41 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5591156 0.90 CTSS (0.56) CTSLCTSBCTSSCTSKWNT1
SCHEMBL5591406 0.83 CTSS (0.63) CTSLCTSBCTSSCTSKWNT1
SCHEMBL5590944 0.81 CTSS (0.68) CTSLCTSBCTSSCTSKMBTD1
SCHEMBL8241923 0.79 CTSL (0.51) CTSLCTSBCTSSCTSKHDAC1
SCHEMBL3165237 0.79 CTSS (0.53) CTSLCTSBCTSSCTSKWNT1
SCHEMBL3159740 0.78 CTSS (0.52) CTSLCTSBCTSSCTSKWNT1
SCHEMBL5591180 0.78 CTSS (0.68) CTSLCTSBCTSSCTSKMBTD1
Trifluoroacetic Acid SCHEMBL5591334 0.77 CTSS (0.62) CTSLCTSBCTSSCTSKHDAC6
SCHEMBL13423600 0.76 CTSL (0.39) CTSLCTSBCTSSCTSKMBTD1
Trifluoroacetic Acid SCHEMBL3175934 0.75 CTSS (0.49) CTSLCTSBCTSSCTSKWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed