SCHEMBL5591269

SCHEMBL5591269

N#Cc1ncc(Br)c(N(CC2CCCC2)NC(=O)c2ccc(CN3CCC(N4CCOCC4)CC3)cc2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.57
CTSS P25774 2/20 0.57
CTSK P43235 2/20 0.57
CTSB P07858 1/20 0.57
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ACVR1 Q04771 4/20 0.40
HRH3 Q9Y5N1 4/20 0.39
CXCR3 P49682 2/20 0.38
BMPR1B O00238 1/20 0.37
BMPR1A P36894 1/20 0.37
TGFBR1 P36897 1/20 0.37
ACVRL1 P37023 1/20 0.37
JAK2 O60674 2/20 0.37
JAK1 P23458 2/20 0.37
JAK3 P52333 2/20 0.37
MBTD1 Q05BQ5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5590944 0.91 CTSS (0.68) CTSLCTSSCTSKCTSBHRH3
SCHEMBL5591180 0.90 CTSS (0.68) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL5591897 0.90 CTSL (0.46) CTSLCTSSCTSKCTSBACVR1
SCHEMBL3159657 0.89 CTSL (0.54) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL5591383 0.89 CTSL (0.63) CTSLCTSSCTSKCTSB
SCHEMBL3159702 0.88 CTSS (0.53) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL5591422 0.88 CTSL (0.62) CTSLCTSSCTSKCTSB
Trifluoroacetic Acid SCHEMBL5591334 0.87 CTSS (0.62) CTSLCTSSCTSKCTSBHRH3
SCHEMBL5590923 0.87 CTSL (0.60) CTSLCTSSCTSKCTSBHRH3
SCHEMBL5591423 0.86 CTSS (0.76) CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed