SCHEMBL5591897

SCHEMBL5591897

N#Cc1ncc(Br)c(N(CC2CCCC2)NC(=O)c2ccc(F)c(CN3CCC(N4CCOCC4)CC3)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSL P07711 6/20 0.46
CTSS P25774 2/20 0.46
CTSK P43235 2/20 0.46
CTSB P07858 1/20 0.46
JAK2 O60674 3/20 0.36
JAK1 P23458 3/20 0.36
JAK3 P52333 3/20 0.36
DDR1 Q08345 2/20 0.35
CXCR3 P49682 2/20 0.34
CCR3 P51677 2/20 0.33
ACVR1 Q04771 2/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
PIK3CG P48736 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5591222 0.96 CTSL (0.43) CTSLCTSSCTSKCTSBJAK2
SCHEMBL8245495 0.94 CTSL (0.47) CTSLCTSSCTSKCTSBCXCR3
SCHEMBL5591269 0.90 CTSL (0.57) CTSLCTSSCTSKCTSBJAK2
SCHEMBL5591381 0.87 CTSL (0.60) CTSLCTSSCTSKCTSBDDR1
Trifluoroacetic Acid SCHEMBL5591672 0.84 CTSS (0.56) CTSLCTSSCTSKCTSB
SCHEMBL5592747 0.82 CTSL (0.52) CTSLCTSSCTSKCTSBJAK2
SCHEMBL5590944 0.81 CTSS (0.68) CTSLCTSSCTSKCTSBCXCR3
SCHEMBL5591156 0.80 CTSS (0.56) CTSLCTSSCTSKCTSBCXCR3
SCHEMBL5591180 0.80 CTSS (0.68) CTSLCTSSCTSKCTSBCXCR3
Trifluoroacetic Acid SCHEMBL5592940 0.79 CTSL (0.48) CTSLCTSSCTSKCTSBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed