SCHEMBL5591383

SCHEMBL5591383

N#Cc1ncc(Br)c(N(CC2CCCC2)NC(=O)c2ccc(CN3CCC(O)CC3)cc2)n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.63
CTSS P25774 2/20 0.63
CTSK P43235 2/20 0.63
CTSB P07858 1/20 0.63
F10 P00742 1/20 0.38
PRKAA2 P54646 10/20 0.38
PRKAB2 O43741 4/20 0.37
PRKAG1 P54619 4/20 0.37
PRKAA1 Q13131 4/20 0.37
PRKAG3 Q9UGI9 4/20 0.37
PRKAG2 Q9UGJ0 4/20 0.37
PRKAB1 Q9Y478 4/20 0.37
HTR2C P28335 1/20 0.36
MCHR1 Q99705 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CHEK1 O14757 1/20 0.36
ACHE P22303 1/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5591343 0.95 CTSL (0.57) CTSLCTSSCTSKCTSBF10
SCHEMBL5591422 0.93 CTSL (0.62) CTSLCTSSCTSKCTSBPRKAA2
SCHEMBL5590923 0.91 CTSL (0.60) CTSLCTSSCTSKCTSBPRKAA2
SCHEMBL5591423 0.91 CTSS (0.76) CTSLCTSSCTSKCTSBF10
SCHEMBL5591580 0.91 CTSS (0.65) CTSLCTSSCTSKCTSBPRKAA2
SCHEMBL8242547 0.90 CTSL (0.51) CTSLCTSSCTSKCTSBF10
SCHEMBL5590919 0.90 CTSS (0.61) CTSLCTSSCTSKCTSBPRKAA2
SCHEMBL5591425 0.90 CTSS (0.67) CTSLCTSSCTSKCTSBPRKAA2
SCHEMBL5591269 0.89 CTSL (0.57) CTSLCTSSCTSKCTSB
SCHEMBL5590944 0.89 CTSS (0.68) CTSLCTSSCTSKCTSBPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed