SCHEMBL5591574

SCHEMBL5591574

CN1CCN(Cc2ccc(-c3cncc(C(=O)NN(CC4CCCC4)c4nc(C#N)ncc4Br)c3)cc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.63
CTSK P43235 5/20 0.63
CTSL P07711 4/20 0.63
CTSB P07858 1/20 0.63
GSK3B P49841 1/20 0.39
DYRK1A Q13627 1/20 0.39
TNIK Q9UKE5 6/20 0.38
MAP3K11 Q16584 1/20 0.37
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37
CHKA P35790 2/20 0.37
TBK1 Q9UHD2 1/20 0.37
EGFR P00533 1/20 0.36
AXL P30530 1/20 0.36
MERTK Q12866 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8245158 0.92 CTSS (0.52) CTSSCTSKCTSLCTSBGSK3B
SCHEMBL5591423 0.91 CTSS (0.76) CTSSCTSKCTSLCTSBCHKA
SCHEMBL3172737 0.89 CTSS (0.59) CTSSCTSKCTSLCTSBGSK3B
SCHEMBL5591471 0.86 CTSS (0.69) CTSSCTSKCTSLCTSBKLKB1
SCHEMBL5591406 0.86 CTSS (0.63) CTSSCTSKCTSLCTSBGSK3B
Trifluoroacetic Acid SCHEMBL5591441 0.86 CTSS (0.69) CTSSCTSKCTSLCTSBTBK1
Trifluoroacetic Acid SCHEMBL3159660 0.85 CTSS (0.55) CTSSCTSKCTSLCTSBGSK3B
SCHEMBL5591180 0.85 CTSS (0.68) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5590944 0.85 CTSS (0.68) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5591415 0.85 CTSS (0.67) CTSSCTSKCTSLCTSBKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed