SCHEMBL5591982

SCHEMBL5591982

N#Cc1ccc(-c2cc(Cl)cc(CCBr)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.42
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP19A1 P11511 2/20 0.38
MMP3 P08254 1/20 0.38
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
KIF11 P52732 2/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585822 0.87 MMP3 (0.40) HRH3TSHRHSD17B10CYP19A1MMP3
SCHEMBL5592063 0.84 MMP3 (0.42) HRH3TSHRHSD17B10CYP19A1MMP3
SCHEMBL3585839 0.81 FFAR4 (0.45) TSHRHSD17B10CYP19A1MMP3MAOA
SCHEMBL27851616 0.80 ADRA1D (0.39) MAOAMAOB
SCHEMBL7275905 0.79 TSHR (0.58) HRH3TSHRHSD17B10CYP19A1MMP3
SCHEMBL16918828 0.79 MMP3 (0.52) TSHRMMP3MAOAMAOBRXRA
SCHEMBL14884590 0.76 CHKA (0.50) HRH3MAOBRXRARXRB
SCHEMBL21302775 0.76 GRM5 (0.51) CYP19A1MMP3MAOAMAOBKIF11
SCHEMBL21313408 0.75 MMP3 (0.44) TSHRMMP3MAOAMAOBRXRA
SCHEMBL508063 0.73 LOXL2 (0.54) TSHRHSD17B10CYP19A1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed