SCHEMBL5592063

SCHEMBL5592063

N#Cc1ccc(-c2cc(Cl)cc(CCO)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.42
HRH3 Q9Y5N1 8/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP19A1 P11511 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
PLAU P00749 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
HSD11B1 P28845 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585839 0.87 FFAR4 (0.45) MMP3TSHRHSD17B10CYP19A1FFAR4
SCHEMBL5591982 0.84 HRH3 (0.42) MMP3HRH3TSHRHSD17B10CYP19A1
SCHEMBL3585822 0.81 MMP3 (0.40) MMP3HRH3TSHRHSD17B10CYP19A1
SCHEMBL8409282 0.79 TSHR (0.58) MMP3HRH3TSHRHSD17B10CYP19A1
SCHEMBL16918828 0.79 MMP3 (0.52) MMP3TSHRRXRARXRBMAOA
SCHEMBL1641272 0.76 HRH3 (0.67) HRH3
SCHEMBL7700731 0.76 CHKA (0.50) TSHRFFAR4RXRARXRBMAOB
SCHEMBL21302775 0.76 GRM5 (0.51) MMP3CYP19A1MAOAMAOB
SCHEMBL320278 0.73 LOXL2 (0.54) TSHRHSD17B10CYP19A1MMP12MMP13
SCHEMBL3598109 0.72 MMP3 (0.42) MMP3HRH3MMP13HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed