SCHEMBL8409282

SCHEMBL8409282

N#Cc1ccc(-c2ccc(CCO)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
HSD17B10 Q99714 1/20 0.58
MMP3 P08254 1/20 0.54
MMP12 P39900 1/20 0.53
MMP13 P45452 1/20 0.53
KCNJ1 P48048 1/20 0.48
KCNH2 Q12809 1/20 0.48
LOXL2 Q9Y4K0 2/20 0.48
CYP2A6 P11509 1/20 0.48
CA2 P00918 1/20 0.46
HRH3 Q9Y5N1 2/20 0.45
KDM1A O60341 1/20 0.44
CYP19A1 P11511 1/20 0.44
KIF11 P52732 2/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320278 0.94 LOXL2 (0.54) TSHRHSD17B10MMP12MMP13KCNJ1
SCHEMBL10773059 0.88 TSHR (0.64) TSHRHSD17B10MMP3MMP12MMP13
SCHEMBL1641272 0.84 HRH3 (0.67) HRH3
Phosphoric Acid SCHEMBL29140249 0.84 KCNJ1 (0.46) TSHRHSD17B10MMP12MMP13KCNJ1
Sulfuric Acid SCHEMBL27373728 0.84 CA2 (0.48) TSHRHSD17B10MMP12MMP13KCNJ1
SCHEMBL17857810 0.83 TSHR (0.72) TSHRHSD17B10MMP3MMP12MMP13
SCHEMBL3236728 0.83 MMP3 (0.58) TSHRHSD17B10MMP3MMP12MMP13
SCHEMBL12807987 0.83 MMP3 (0.58) TSHRHSD17B10MMP3MMP12MMP13
SCHEMBL2771783 0.82 MMP12 (0.59) MMP12MMP13HDAC8
SCHEMBL2044945 0.82 CA2 (0.65) TSHRCA2HRH3MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed