SCHEMBL5595477

SCHEMBL5595477

CC=C(O[Si](C)(C)C)c1ccc(OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
CES2 O00748 2/20 0.45
CES1 P23141 2/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
CA1 P00915 6/20 0.44
CA2 P00918 6/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
NR1I2 O75469 1/20 0.42
PARP1 P09874 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
PARP4 Q9UKK3 1/20 0.42
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5595475 1.00 PRSS1 (0.47) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL13811105 0.84 KDM4E (0.51) ALDH1A1KDM4EHPGDCYP2C19HSD17B10
SCHEMBL13811104 0.80 ALDH1A1 (0.39) CES2CES1ALDH1A1KDM4EMAPT
SCHEMBL2091071 0.79 CA1 (0.54) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL8742243 0.78 LMNA (0.38) CES2CES1ALDH1A1MAPTHPGD
SCHEMBL13245881 0.78 LMNA (0.38) CES2CES1ALDH1A1MAPTHPGD
SCHEMBL817341 0.78 TSHR (0.35) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL4442135 0.78 TSHR (0.35) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL5595601 0.78 TSHR (0.35) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL23152625 0.76 SMN1; SMN2 (0.42) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203616-B1 CHIRAL LEAD CATALYST AND METHOD OF ASYMMETRIC ALDOL REACTION JAPAN SCIENCE & TECH AGENCY (JP) 2007-01-10 EP disclosed
US-6780812-B2 SUCH AS LEAD TRIFLATE AND A CHIRAL CROWN ETHER COMPOUND JAPAN SCIENCE AND TECHNOLOGY CORPORATION (JP) 2004-08-24 US disclosed
US-20040087437-A1 CHIRAL LEAD CATALYST AND METHOD OF ASYMMETRIC ALDOL REACTION JAPAN SCIENCE AND TECHNOLOGY CORPORATION (JP) 2004-05-06 US disclosed
EP-1203616-A1 CHIRAL LEAD CATALYST AND METHOD OF ASYMMETRIC ALDOL REACTION Japan Science and Technology Corporation (JP) 2002-05-08 EP disclosed