SCHEMBL5596130

SCHEMBL5596130

[c]1nc(N2CCN(c3cnccn3)CC2)ncc1-c1nc2ccccc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.44
AURKA O14965 1/20 0.41
FLT4 P35916 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
SORD Q00796 2/20 0.39
LMNA P02545 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DRD2 P14416 6/20 0.38
HTR1A P08908 5/20 0.38
HTR7 P34969 5/20 0.38
DRD4 P21917 4/20 0.38
DRD3 P35462 4/20 0.38
HTR2A P28223 4/20 0.38
ADRA2A P08913 2/20 0.38
ADRA2C P18825 2/20 0.38
SLC6A2 P23975 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5596399 0.87 HTR1A (0.48) IRAK4AURKAFLT4NPC1RAB9A
SCHEMBL5596653 0.73 SCD (0.42) NPC1RAB9AALDH1A1TSHRLMNA
SCHEMBL4949763 0.68 MAPK8 (0.41) IRAK4AURKAFLT4NPC1RAB9A
SCHEMBL4023738 0.67 MAPK10 (0.56) IRAK4NPC1RAB9AALDH1A1TSHR
SCHEMBL219434 0.67 NPC1 (0.67) NPC1RAB9AALDH1A1TSHRHSD17B10
SCHEMBL29373464 0.67 NPC1 (0.67) NPC1RAB9AALDH1A1TSHRHSD17B10
SCHEMBL5596467 0.67 NPC1 (0.48) NPC1RAB9AALDH1A1TSHRHSD17B10
SCHEMBL5596753 0.67 ILK (0.56) NPC1RAB9AALDH1A1L3MBTL1KDM4E
SCHEMBL5564234 0.66 SORD (0.43) IRAK4NPC1RAB9AALDH1A1TSHR
SCHEMBL5596604 0.65 ILK (0.52) IRAK4RAB9ATSHRTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696909-B1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES SERONO LAB (CH) 2007-11-14 EP claimed