SCHEMBL5596256

SCHEMBL5596256

[c]1nc(NCCc2ccccc2)ncc1-c1nc2ccccc2s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ILK Q13418 2/20 0.42
APP P05067 3/20 0.41
CDK1 P06493 1/20 0.41
KDR P35968 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5596937 0.91 ILK (0.53) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596418 0.91 NPC1 (0.44) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596939 0.91 NPC1 (0.44) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596674 0.91 NPC1 (0.44) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596411 0.91 RAB9A (0.45) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5597099 0.88 PTGS1 (0.46) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596896 0.88 CSNK1D (0.45) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5597098 0.87 MAPT (0.49) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL5596261 0.86 ALDH1A1 (0.44) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL5596942 0.85 ILK (0.51) NPC1RAB9AALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696909-B1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES SERONO LAB (CH) 2007-11-14 EP claimed