SCHEMBL5596285

SCHEMBL5596285

[c]1nc(NCc2ccccn2)ncc1-c1nc2ccccc2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.47
NPC1 O15118 5/20 0.47
RAB9A P51151 5/20 0.47
ALDH1A1 P00352 4/20 0.47
TP53 P04637 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HSD17B10 Q99714 2/20 0.47
TSHR P16473 2/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
HTT P42858 2/20 0.42
HPGD P15428 1/20 0.42
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5596753 0.82 ILK (0.56) KDM4ENPC1RAB9AALDH1A1CCNE1
SCHEMBL5596344 0.81 RAB9A (0.46) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596942 0.80 ILK (0.51) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596256 0.79 NPC1 (0.54) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596406 0.78 ILK (0.51) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596435 0.78 ILK (0.40) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596495 0.76 LTA4H (0.39) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596674 0.76 NPC1 (0.44) NPC1RAB9AALDH1A1SMN1; SMN2HTT
SCHEMBL5596418 0.76 NPC1 (0.44) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5596937 0.76 ILK (0.53) KDM4ENPC1RAB9AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696909-B1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES SERONO LAB (CH) 2007-11-14 EP claimed