SCHEMBL5599336

SCHEMBL5599336

Cn1cc(Cc2ccc(OCCC(Cl)N3CCCC3)cc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.45
PSMB5 P28074 1/20 0.45
PSMB2 P49721 1/20 0.45
LTA4H P09960 13/20 0.44
HRH3 Q9Y5N1 4/20 0.44
TSHR P16473 1/20 0.38
ACHE P22303 1/20 0.38
RAD52 P43351 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599425 0.77 PSMB1 (0.43) PSMB1PSMB5PSMB2LTA4HHRH3
SCHEMBL5599288 0.73 PSMB1 (0.36) PSMB1PSMB5PSMB2LTA4HHRH3
SCHEMBL5611378 0.70 LTA4H (0.34) PSMB1PSMB5PSMB2LTA4HHRH3
SCHEMBL25680303 0.68 KCNH2 (0.56) LTA4H
SCHEMBL30628842 0.67 KCNH2 (0.43)
SCHEMBL16877094 0.64 CALM1 (0.48) LTA4H
SCHEMBL25902251 0.63 TDP1 (0.49)
SCHEMBL7134872 0.62 LTA4H (1.00) PSMB1PSMB5PSMB2LTA4HHRH3
SCHEMBL9527901 0.61 HRH3 (0.74) PSMB1PSMB5PSMB2LTA4HHRH3
SCHEMBL7139563 0.61 LTA4H (1.00) PSMB1PSMB5PSMB2LTA4HHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1746986-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-01-31 EP claimed
WO-2005097099-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO claimed
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed